SCHEMBL22809481

SCHEMBL22809481

CNCCOc1ccc2cc(C(F)(F)F)ccc2n1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
SCN9A Q15858 13/20 0.44
SCN10A Q9Y5Y9 2/20 0.43
RAF1 P04049 1/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE7A Q13946 1/20 0.40
SCN7A Q01118 3/20 0.39
KCNH2 Q12809 3/20 0.39
SCN5A Q14524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809472 0.82 BACE1 (0.54) BACE1SCN9ASCN10APDE1APDE1B
Hydrochloric Acid SCHEMBL20595231 0.81 BACE1 (0.53) BACE1SCN9ASCN10APDE1APDE1B
SCHEMBL28354796 0.80 SCN9A (0.48) SCN9ASCN10ASCN7AKCNH2SCN5A
SCHEMBL28350726 0.75 BACE1 (0.47) BACE1SCN9ASCN10APDE1APDE1B
SCHEMBL30465758 0.75 MAPT (0.56)
SCHEMBL22809595 0.75 BACE1 (0.49) BACE1SCN9A
SCHEMBL22809583 0.74 BACE1 (0.41) BACE1SCN9ASCN10APDE1APDE1B
SCHEMBL167871 0.74 HTR1B (0.49) KCNH2
SCHEMBL22809542 0.73 RXFP1 (0.44) RAF1KCNH2
SCHEMBL22809568 0.71 L3MBTL4 (0.52) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed