SCHEMBL22809607

SCHEMBL22809607

Cc1cc(C(F)(F)F)cnc1O[C@H](C)CN

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGS2 P35354 4/20 0.37
SSTR4 P31391 1/20 0.37
NPSR1 Q6W5P4 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SCN9A Q15858 1/20 0.34
KMT2A Q03164 3/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 2/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809491 0.85 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL22809492 0.85 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL22809475 0.85 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL28354502 0.84 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL28354503 0.84 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL28354724 0.84 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL17055785 0.79 AGBL2 (0.41) AGBL2CYP1A2CYP3A4CYP2C19PTGS2
SCHEMBL17055784 0.74 PTGS2 (0.52) AGBL2CYP1A2CYP3A4CYP2C19PTGS2
SCHEMBL18312359 0.74 NPSR1 (0.47) AGBL2CYP1A2CYP3A4CYP2C19PTGS2
SCHEMBL8427120 0.73 KMT2A (0.47) AGBL2CYP1A2CYP3A4CYP2C19PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed