SCHEMBL22809647

SCHEMBL22809647

CC(F)(F)Oc1ccc(OCCN)cc1F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.42
PDK2 Q15119 2/20 0.41
SLC7A5 Q01650 1/20 0.40
LTA4H P09960 2/20 0.39
PDE2A O00408 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
PLA2G2A P14555 1/20 0.38
FFAR1 O14842 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
ESR1 P03372 1/20 0.35
CYP19A1 P11511 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809574 0.87 SLC7A5 (0.50) SMN1; SMN2PDK2SLC7A5LTA4HPDE2A
Hydrochloric Acid SCHEMBL28350715 0.86 SLC7A5 (0.49) SMN1; SMN2PDK2SLC7A5LTA4HPDE2A
Hydrochloric Acid SCHEMBL30450035 0.86 SLC7A5 (0.49) SMN1; SMN2PDK2SLC7A5LTA4HPDE2A
SCHEMBL1683223 0.76 SMN1; SMN2 (0.45) SMN1; SMN2PDK2SLC7A5LTA4HTAAR1
SCHEMBL26334840 0.75 PPARD (0.41) SLC7A5FFAR1PPARGPPARD
SCHEMBL18295348 0.74 TAAR1 (0.47) SMN1; SMN2PDK2LTA4HTAAR1PLA2G2A
SCHEMBL25799178 0.74 S1PR4 (0.40) PDK2FFAR1PPARGPPARD
SCHEMBL26334630 0.74 S1PR4 (0.40) PDK2FFAR1PPARGPPARD
SCHEMBL4856586 0.74 MAOB (0.54) SMN1; SMN2PDK2LTA4HTAAR1PLA2G2A
SCHEMBL22809630 0.73 SLC7A5 (0.48) SMN1; SMN2PDK2SLC7A5LTA4HTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed