SCHEMBL22809689

SCHEMBL22809689

CC(C)CCOc1cc(C(F)(F)F)ccc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 2/20 0.48
SCN10A Q9Y5Y9 2/20 0.48
TRPV1 Q8NER1 1/20 0.42
ALDH1A1 P00352 6/20 0.40
HTT P42858 4/20 0.40
HPGD P15428 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.40
MAPT P10636 1/20 0.40
ESR1 P03372 1/20 0.40
TLR8 Q9NR97 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HSD17B10 Q99714 2/20 0.38
USP2 O75604 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809662 0.87 SCN8A (0.46) SCN8ASCN10ATRPV1ALDH1A1HTT
SCHEMBL955509 0.85 CYP1A1 (0.46) SCN8ASCN10ATRPV1ALDH1A1HTT
SCHEMBL953869 0.84 PTGDR2 (0.48) ALDH1A1HTTHPGDSMN1; SMN2POLB
SCHEMBL22090766 0.83 KDM4E (0.45) SCN8ASCN10AALDH1A1HTTHPGD
SCHEMBL31136545 0.82 ALDH1A1 (0.42) SCN8ASCN10AALDH1A1HTTHPGD
SCHEMBL957465 0.82 CYP2C19 (0.50) ALDH1A1HPGDPOLBMAPTKDM4E
SCHEMBL28639293 0.81 ALDH1A1 (0.47) ALDH1A1HTTHPGDSMN1; SMN2MAPT
SCHEMBL21722870 0.80 APP (0.46) ALDH1A1HTTHPGDSMN1; SMN2POLB
SCHEMBL22432922 0.80 POLB (0.39) SCN8ASCN10ATRPV1ALDH1A1HTT
SCHEMBL22090747 0.79 POLB (0.41) ALDH1A1HTTHPGDSMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3239134-B1 PYRIDONE AMIDES AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2020-12-23 EP disclosed