SCHEMBL22818975

SCHEMBL22818975

Cc1ccc(C2=N/C(=C\c3ccc(F)cc3)CO2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.45
NFE2L2 Q16236 1/20 0.42
PTGS1 P23219 1/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
ALOX5 P09917 1/20 0.38
ACHE P22303 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAOB P27338 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
RECQL P46063 1/20 0.33
MDM2 Q00987 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
AR P10275 1/20 0.33
MAPK1 P28482 1/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22818979 0.70 MAPK1 (0.64) RAB9ANPC1ALOX5ALDH1A1KDM4E
SCHEMBL66437 0.66 PTGS1 (0.42) RAB9APTGS1MAPTNPC1HTT
SCHEMBL29727510 0.66 NFE2L2 (0.51) NFE2L2MAPTALDH1A1MAOB
SCHEMBL10630404 0.65 KMT2A (0.50) RAB9APTGS1MAPTNPC1HTT
SCHEMBL20804472 0.63 ACHE (0.81) RAB9ANFE2L2PTGS1NPC1ACHE
SCHEMBL422511 0.63 ACHE (0.81) RAB9ANFE2L2PTGS1NPC1ACHE
SCHEMBL29693877 0.63 APP (0.40) MAPTHTTALOX5MAOB
SCHEMBL11532298 0.62 NFE2L2 (1.00) NFE2L2PTGS1ALOX5ACHE
SCHEMBL18240780 0.62 NFE2L2 (0.73) RAB9ANFE2L2PTGS1NPC1ALOX5
SCHEMBL11532304 0.62 NFE2L2 (1.00) NFE2L2PTGS1ALOX5ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020257790-A1 PHARMACEUTICALLY ACTIVE PYRAZOLO-PYRIDONE MODULATORS OF DCN1/2-MEDIATED CULLIN NEDDYLATION UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2020-12-24 WO disclosed