SCHEMBL2283129

SCHEMBL2283129

Cc1cc(C)cc(CC(N)c2cnn(C)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.35
LRRK2 Q5S007 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
AXL P30530 1/20 0.32
MERTK Q12866 1/20 0.32
OPRM1 P35372 1/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
ACLY P53396 1/20 0.31
MPO P05164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
FYN P06241 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12706271 0.75 TACR1 (0.44) TACR1NOS1NOS2ALDH1A1
SCHEMBL17018452 0.74 SLC6A4 (0.37) LRRK2OPRM1MPOALDH1A1HTT
SCHEMBL16447921 0.74 IDO1 (0.32) LRRK2OPRM1MPOALDH1A1HTT
SCHEMBL3466744 0.74 SLC6A4 (0.37) LRRK2OPRM1MPOALDH1A1HTT
SCHEMBL18793288 0.73 SMN1; SMN2 (0.34) OPRM1MPOALDH1A1LMNAHTT
Hydrochloric Acid SCHEMBL27164845 0.73 SLC6A4 (0.36) OPRM1ALDH1A1HTT
SCHEMBL2289154 0.71
SCHEMBL3924798 0.69 TACR1 (0.44) TACR1NOS1NOS2LMNAMAPT
SCHEMBL28802900 0.68
SCHEMBL2303823 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989394-B2 Substituted 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds BASF SE (DE) 2011-08-02 US disclosed
US-20090131256-A1 Substituted 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane Compounds BASF SE (DE) 2009-05-21 US disclosed
EP-2041089-A1 SUBSTITUTED 1-(AZOLIN-2-YL)-AMINO-2-ARYL-1-HETARYL-ETHANE COMPOUNDS BASF SE (DE) 2009-04-01 EP disclosed
WO-2008000834-A1 SUBSTITUTED 1-(AZOLIN-2-YL)-AMINO-2-ARYL-1-HETARYL-ETHANE COMPOUNDS BASF SE (DE) 2008-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090131256-A1 Substituted 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane Compounds AAAS, AIPL1, ATXN2 TACR1 1143/4885LRRK2 2897/4885CYP11B1 1601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.