SCHEMBL22838720

SCHEMBL22838720

CNc1cc(-c2ccc(F)nc2)ncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.46
CLK4 Q9HAZ1 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP2D6 P10635 3/20 0.46
HSD17B10 Q99714 3/20 0.46
ALOX15 P16050 2/20 0.46
CYP3A4 P08684 3/20 0.46
SYK P43405 2/20 0.44
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK1 P28482 1/20 0.42
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
MAPT P10636 5/20 0.41
CYP2A6 P11509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905207 0.82 CYP1A2 (0.51) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL20816287 0.81 CYP1A2 (0.58) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL28017373 0.80 ABL1 (0.55) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL28017385 0.79 ABL1 (0.54) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL15933190 0.78 MAPT (0.49) CLK4CYP2C19CYP3A4SYKMAPT
SCHEMBL22838692 0.77 CYP1A2 (0.43) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL22838564 0.76 CYP1A2 (0.51) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL22838698 0.76 SYK (0.42) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL16373642 0.75 CYP1A2 (0.50) CYP1A2CLK4CYP2C19CYP2D6HSD17B10
SCHEMBL20816288 0.75 FAAH (0.51) CYP1A2CLK4CYP2C19CYP2D6HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3459942-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2020-12-30 EP disclosed