SCHEMBL22838698

SCHEMBL22838698

CNc1cc(-c2ccc(C(C)(C)O)nc2)ncn1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SYK P43405 12/20 0.42
CYP1A2 P05177 4/20 0.42
CLK4 Q9HAZ1 2/20 0.42
CYP2D6 P10635 2/20 0.42
HSD17B10 Q99714 2/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYP3A4 P08684 1/20 0.42
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
JAK2 O60674 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28017373 0.84 ABL1 (0.55) CYP1A2CLK4CYP2D6HSD17B10ALOX15
Hydrochloric Acid SCHEMBL28017385 0.83 ABL1 (0.54) CYP1A2CLK4CYP2D6HSD17B10ALOX15
SCHEMBL15473171 0.82 FAAH (0.47) SYK
SCHEMBL19905207 0.77 CYP1A2 (0.51) CYP1A2CLK4CYP2D6HSD17B10ALOX15
SCHEMBL22838720 0.76 CYP1A2 (0.46) SYKCYP1A2CLK4CYP2D6HSD17B10
SCHEMBL16664930 0.73 GPR39 (0.42) CYP1A2CLK4CYP2D6HSD17B10ALOX15
SCHEMBL22838692 0.72 CYP1A2 (0.43) CYP1A2CLK4CYP2D6HSD17B10ALOX15
SCHEMBL22838564 0.72 CYP1A2 (0.51) CYP1A2CLK4CYP2D6HSD17B10ALOX15
SCHEMBL16660252 0.70 FAAH (0.49)
SCHEMBL16373642 0.70 CYP1A2 (0.50) CYP1A2CLK4CYP2D6HSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3459942-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2020-12-30 EP disclosed