SCHEMBL22844183

SCHEMBL22844183

CC(C)(C)[Si](C)(C)OCCC[C@H](Cn1c(N)nc2ccccc21)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 4/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
HTT P42858 1/20 0.39
CXCR4 P61073 1/20 0.39
TLR8 Q9NR97 3/20 0.39
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TNF P01375 1/20 0.36
CXCL8 P10145 1/20 0.36
SOS1 Q07889 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
F2R P25116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22844249 0.83 HTT (0.45) CYP1A2CYP2D6HTTCXCR4TLR8
SCHEMBL2031432 0.78 CXCR4 (0.62) CYP1A2CYP2D6HTTCXCR4TLR8
SCHEMBL22844182 0.76 CXCR4 (0.63) CYP1A2CYP2D6HTTCXCR4TLR8
SCHEMBL6939027 0.71 ADA (0.40)
SCHEMBL8440133 0.69 CETP (0.36)
SCHEMBL14587571 0.69 TBXAS1 (0.45) L3MBTL1
SCHEMBL22844244 0.67 CASR (0.39) CSF1RTLR8POLB
SCHEMBL31411073 0.67 BTN3A1 (0.35) CYP1A2CYP2D6HTTMEN1KMT2A
SCHEMBL13219003 0.66 BTN3A1 (0.35)
SCHEMBL20769894 0.65 SMN1; SMN2 (0.52) HTTPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020260252-A1 NEW MACROCYCLIC COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-12-30 WO disclosed