SCHEMBL22844244

SCHEMBL22844244

COc1cccc2nc(N)n(C[C@H](C)CCCO[Si](C)(C)C(C)(C)C)c12

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASR P41180 3/20 0.39
TLR8 Q9NR97 2/20 0.36
CSF1R P07333 2/20 0.32
DCPS Q96C86 3/20 0.32
NQO2 P16083 3/20 0.32
DHFR P00374 2/20 0.32
POLB P06746 2/20 0.31
DUT P33316 1/20 0.30
LMNA P02545 2/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
G6PD P11413 1/20 0.30
PKM P14618 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22844249 0.82 HTT (0.45) TLR8POLBLMNA
SCHEMBL2031432 0.68 CXCR4 (0.62) TLR8POLBLMNANPC1RAB9A
SCHEMBL22844246 0.68 DRD3 (0.37) NPC1RAB9A
SCHEMBL22844183 0.67 CSF1R (0.41) TLR8CSF1RPOLB
SCHEMBL22844182 0.66 CXCR4 (0.63) TLR8POLBMAPT
SCHEMBL22844210 0.65 DUT (0.34) DUT
SCHEMBL6530152 0.64 CYP2D6 (0.50) POLBLMNAMAPT
SCHEMBL6606918 0.64 LMNA (0.41) LMNANPC1MAPTPKMRAB9A
SCHEMBL22571857 0.63 STING1 (0.41) NPC1RAB9A
SCHEMBL5459067 0.63 PRMT5 (0.60) CASRTLR8DCPSNQO2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020260252-A1 NEW MACROCYCLIC COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-12-30 WO disclosed