SCHEMBL22848331

SCHEMBL22848331

CNC(=O)c1cc(F)c(-c2c(N)cccc2F)nc1N(C=O)c1c(CCC(=O)O)ccnc1C(C)C

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 13/20 0.36
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
ALOX5AP P20292 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22848185 0.86 KRAS (0.34) KRAS
SCHEMBL24372814 0.71 KRAS (0.35) KRAS
SCHEMBL26527390 0.71 KRAS (0.42) KRAS
SCHEMBL26036624 0.69 KRAS (0.32) KRAS
SCHEMBL29614930 0.69 KRAS (0.54) KRAS
SCHEMBL24436419 0.69 KRAS (0.54) KRAS
SCHEMBL20805455 0.68 KRAS (0.45) KRAS
SCHEMBL26525295 0.68 KRAS (0.51) KRAS
SCHEMBL22848330 0.68 KRAS (0.41) KRAS
SCHEMBL20805634 0.68 KRAS (0.49) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020259513-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF KRAS G12C GUANGDONG NEWOPP BIOPHARMACEUTICALS CO., LTD. (CN) 2020-12-30 WO disclosed