SCHEMBL22852811

SCHEMBL22852811

CCOC(=O)c1ccc(OC)cc1Nc1ccc(F)cc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.50
P2RX7 Q99572 1/20 0.49
AKR1C3 P42330 6/20 0.45
AKR1C2 P52895 6/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 3/20 0.44
GAA P10253 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 2/20 0.44
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TP53 P04637 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPK14 Q16539 1/20 0.43
MAOB P27338 2/20 0.43
CA12 O43570 1/20 0.43
CA2 P00918 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294267 1.00 CDC25B (0.50) CDC25BP2RX7AKR1C3AKR1C2ALDH1A1
SCHEMBL30294387 0.85 ALDH1A1 (0.44) CDC25BALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL30294718 0.85 AKR1C3 (0.63) AKR1C3AKR1C2
SCHEMBL22853342 0.85 AKR1C3 (0.63) AKR1C3AKR1C2
SCHEMBL22853397 0.84 MAPT (0.49) ALDH1A1KDM4ESMN1; SMN2LMNAPOLB
SCHEMBL30294784 0.84 MAPT (0.49) ALDH1A1KDM4ESMN1; SMN2LMNAPOLB
SCHEMBL22833395 0.82 KDM4E (0.46) KDM4ESMN1; SMN2LMNAPOLBTDP1
SCHEMBL29382578 0.82 KDM4E (0.46) KDM4ESMN1; SMN2LMNAPOLBTDP1
SCHEMBL10834109 0.81 CDC25B (0.65) CDC25BP2RX7AKR1C3AKR1C2ALDH1A1
SCHEMBL22853336 0.81 SMN1; SMN2 (0.42) ALDH1A1HPGDKDM4EGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed