SCHEMBL22852994

SCHEMBL22852994

Cc1ccc(Nc2ccc(F)cc2C)c(C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 14/20 0.56
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPK1 P28482 1/20 0.52
FABP3 P05413 2/20 0.50
FABP4 P15090 2/20 0.50
P2RY4 P51582 1/20 0.50
GFER P55789 1/20 0.48
AKR1C3 P42330 1/20 0.47
AKR1C2 P52895 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294529 1.00 DHODH (0.56) DHODHMEN1KMT2AMAPK1FABP3
SCHEMBL30294653 0.92 P2RY4 (0.56) DHODHMEN1KMT2AMAPK1FABP3
SCHEMBL22853383 0.92 P2RY4 (0.56) DHODHMEN1KMT2AMAPK1FABP3
SCHEMBL22852993 0.85 KDM4E (0.54) DHODHMEN1KMT2AFABP3FABP4
SCHEMBL30294397 0.85 KDM4E (0.54) DHODHMEN1KMT2AFABP3FABP4
SCHEMBL22853121 0.85 IDO1 (0.48) DHODHMEN1KMT2AMAPK1FABP3
SCHEMBL30294377 0.85 IDO1 (0.48) DHODHMEN1KMT2AMAPK1FABP3
SCHEMBL22853331 0.85 AKR1C3 (0.59) MEN1KMT2AMAPK1FABP3FABP4
SCHEMBL30294672 0.85 AKR1C3 (0.59) MEN1KMT2AMAPK1FABP3FABP4
SCHEMBL22853346 0.84 IDO1 (0.50) DHODHMEN1KMT2AMAPK1FABP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed