SCHEMBL22853709

SCHEMBL22853709

COC(=O)C(C)OC(=O)CC[C@@H]1N=C(c2ccccn2)c2cc(Br)ccc2-n2c(C)cnc21

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
BRD4 O60885 2/20 0.35
HDAC6 Q9UBN7 4/20 0.31
HDAC1 Q13547 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22853711 0.94 GABRA5 (0.39) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL18808051 0.92 GABRA1 (0.41) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL18808052 0.92 GABRA1 (0.41) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL22853772 0.92 GABRA1 (0.38) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL22853765 0.92 BRD4 (0.33) BRD4HDAC6HDAC1
Remimazolam SCHEMBL23735014 0.91 GABRA1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
Remimazolam SCHEMBL29579211 0.91 GABRA1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
Remimazolam SCHEMBL846435 0.91 GABRA1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
Remimazolam SCHEMBL29379415 0.91 GABRA1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL22853702 0.90 GABRA1 (0.39) GABRA1GABRA5GABRA3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3992194-A1 BENZODIAZEPINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF IN MEDICINE West China Hospital, Sichuan University (CN) 2022-05-04 EP disclosed
WO-2020259602-A1 BENZODIAZEPINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF IN MEDICINE 四川大学华西医院 2020-12-30 WO disclosed