SCHEMBL22856415

SCHEMBL22856415

CCCCC1CCN(c2ccc(CC(C)(C)C)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.41
HRH3 Q9Y5N1 2/20 0.40
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
S1PR1 P21453 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ESR1 P03372 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
HTR1A P08908 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
CHRM1 P11229 1/20 0.36
DRD2 P14416 1/20 0.36
ADRA2B P18089 1/20 0.36
CHRM3 P20309 1/20 0.36
DRD4 P21917 1/20 0.36
ADRA1D P25100 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30516679 0.86 KDM4E (0.44) DPP4HRH3CYP1A2S1PR1MAOA
SCHEMBL25192949 0.83 MAPT (0.51) DPP4HRH3CYP1A2POLB
SCHEMBL24359587 0.81 HRH3 (0.45) DPP4HRH3S1PR1MAOAMAOB
SCHEMBL23842183 0.81 DPP4 (0.40) DPP4HRH3CYP1A2S1PR1MAOA
SCHEMBL24508492 0.81 RORC (0.40) HRH3ESR1CHRM4
SCHEMBL23696638 0.81 DPP4 (0.40) DPP4HRH3
SCHEMBL15037944 0.80 DPP4 (0.60) DPP4HRH3CHRM2CHRM4HTR1A
SCHEMBL26845651 0.79 ESR1 (0.38) HRH3CYP1A2HPGDESR1
SCHEMBL26845653 0.79 ESR1 (0.38) HRH3CYP1A2HPGDESR1
SCHEMBL22794821 0.76 KDM4E (0.46) HRH3MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020264490-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2020-12-30 WO disclosed