SCHEMBL22868059

SCHEMBL22868059

NC(c1ccc(CC(F)(F)F)cc1)c1ccc(CC(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
PDE2A O00408 6/20 0.33
GRB2 P62993 1/20 0.33
HSD17B2 P37059 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
F2 P00734 1/20 0.31
TAAR1 Q96RJ0 1/20 0.30
SLC6A2 P23975 1/20 0.30
HTR2A P28223 1/20 0.30
SLC6A4 P31645 1/20 0.30
HRH1 P35367 1/20 0.30
HTR2B P41595 1/20 0.30
CHRNA4 P43681 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7670360 0.80 ESR1 (0.38) ESR1ESR2CYP1A2CYP2C19TAAR1
SCHEMBL12050478 0.77 IDO1 (0.47) PDE2ACYP2D6
SCHEMBL10570 0.75 ALDH1A1 (0.52) TAAR1
SCHEMBL22423075 0.75 PDE2A (0.36) ESR1ESR2PDE2AHSD17B2CYP1A2
SCHEMBL18103202 0.74 PTPN5 (0.42) ESR1ESR2PDE2AHSD17B2CYP2C19
SCHEMBL34471882 0.74 TAAR1 (0.55) TAAR1SLC6A2HTR2ASLC6A4HTR2B
SCHEMBL3888293 0.73 LOXL2 (0.55) TAAR1
SCHEMBL8911483 0.72 PDE2A (0.34) ESR1ESR2PDE2AHSD17B2
SCHEMBL18358078 0.72 TSHR (0.42) ESR1ESR2PDE2AGRB2HSD17B2
SCHEMBL20382684 0.71 PDE2A (0.36) ESR1ESR2PDE2AHSD17B2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed