SCHEMBL22868063

SCHEMBL22868063

CC(C)(C)OC(=O)Nc1ccc(CSc2ncc(C(=O)O)c(=O)[nH]2)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 11/20 0.61
KDM4A O75164 11/20 0.61
KDM4D Q6B0I6 11/20 0.61
HIF1AN Q9NWT6 11/20 0.61
KDM2A Q9Y2K7 11/20 0.61
KDM5B Q9UGL1 9/20 0.61
SCN9A Q15858 1/20 0.49
KDM3B Q7LBC6 9/20 0.49
DAO P14920 2/20 0.44
CYP17A1 P05093 1/20 0.43
PLA2G7 Q13093 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
PSMB8 P28062 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22868062 0.88 CA12 (0.47) KDM6BKDM4AKDM4DHIF1ANKDM2A
SCHEMBL29580908 0.78 HSD17B1 (0.46) KDM6BKDM4AKDM4DHIF1ANKDM2A
SCHEMBL22867869 0.78 HSD17B1 (0.46) KDM6BKDM4AKDM4DHIF1ANKDM2A
SCHEMBL22425202 0.72 CYP17A1 (0.58) SCN9ACYP17A1PTGDR2PSMB8
SCHEMBL23092683 0.70 MEN1 (0.53) CYP17A1
SCHEMBL10361607 0.69 CYP17A1 (0.61) CYP17A1PTGDR2PSMB8
SCHEMBL14076457 0.69 CYP17A1 (0.54) SCN9ACYP17A1PTGDR2PSMB8
SCHEMBL132701 0.68 CYP17A1 (0.76) CYP17A1PTGDR2PSMB8
SCHEMBL13055402 0.67 CYP17A1 (0.59) CYP17A1PTGDR2PSMB8
SCHEMBL702839 0.67 CYP17A1 (0.58) CYP17A1PTGDR2PSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994125-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF Regeneron Pharmaceuticals, Inc. (US) 2022-05-11 EP disclosed
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed