SCHEMBL22878342

SCHEMBL22878342

O=C1OCCN1CCCN1C[C@H]2CN(I)C[C@H]2C1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
PIK3CD O00329 1/20 0.33
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
NAAA Q02083 1/20 0.31
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17285928 0.87 KDM4E (0.38) KDM4EPIK3CDCNR1CNR2NAAA
SCHEMBL17284567 0.85 KDM4E (0.38) KDM4EPIK3CDCNR1CNR2NQO2
SCHEMBL17281979 0.82 KDM4E (0.35) KDM4EPIK3CDCNR1CNR2NQO2
SCHEMBL22878344 0.75 ADRA1B (0.41) PIK3CD
SCHEMBL10778747 0.74 HRH3 (0.43) KDM4EPIK3CD
SCHEMBL22878356 0.73 KEAP1 (0.47) KDM4E
SCHEMBL16377754 0.72 KDM4E (0.46) KDM4EPIK3CDCNR1CNR2NAAA
SCHEMBL7625818 0.72 CXCR4 (0.44) KDM4EPIK3CD
SCHEMBL17789613 0.71 PIK3CD (0.50) KDM4EPIK3CDCNR1CNR2NAAA
SCHEMBL18672857 0.70 PIK3CD (0.49) KDM4EPIK3CDCNR1CNR2NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145929-B1 5-CHLORO-2-DIFLUOROMETHOXYPHENYL PYRAZOLOPYRIMIDINE COMPOUNDS WHICH ARE JAK INHIBITORS HOFFMANN LA ROCHE (CH) 2021-01-13 EP disclosed