SCHEMBL22889934

SCHEMBL22889934

COC(=O)c1ncc(Br)c(OC)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.39
PTPN1 P18031 1/20 0.36
HPGD P15428 3/20 0.34
MAPK1 P28482 3/20 0.34
ATM Q13315 2/20 0.34
MAPT P10636 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 2/20 0.33
LMNA P02545 2/20 0.33
GMNN O75496 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
GABRA1 P14867 1/20 0.33
TSHR P16473 1/20 0.33
GABRG2 P18507 1/20 0.33
NFKB1 P19838 1/20 0.33
APEX1 P27695 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29771512 0.85 HSD17B10 (0.41) PTPN1HPGDMAPTALDH1A1KDM4E
SCHEMBL22890254 0.85 HSD17B10 (0.41) PTPN1HPGDMAPTALDH1A1KDM4E
SCHEMBL7665937 0.83 AGXT (0.44) NPSR1HPGDMAPK1ATMMAPT
SCHEMBL22890486 0.79 NPSR1 (0.38) NPSR1HPGDMAPK1ATMMAPT
SCHEMBL22890261 0.78 NPSR1 (0.37) NPSR1HPGDMAPK1ATMMAPT
SCHEMBL9939724 0.77 NPSR1 (0.39) NPSR1PTPN1MAPK1ATMMAPT
SCHEMBL7588137 0.75 NPSR1 (0.45) NPSR1MAPK1ATMMAPTL3MBTL1
SCHEMBL26260299 0.75 HSD17B10 (0.41) PTPN1HPGDMAPTALDH1A1KDM4E
SCHEMBL31500546 0.72 NPSR1 (0.47) NPSR1HPGDMAPK1ATMMAPT
SCHEMBL31184927 0.72 L3MBTL1 (0.46) NPSR1MAPK1L3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021007477-A1 INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2021-01-14 WO disclosed