SCHEMBL22901561

SCHEMBL22901561

COc1cccc(COc2cc(F)cc3ccc(-c4nccc(C)n4)nc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GCK P35557 1/20 0.42
ABCB1 P08183 2/20 0.40
FFAR1 O14842 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
APP P05067 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
F2RL3 Q96RI0 2/20 0.39
MPO P05164 1/20 0.39
SGMS2 Q8NHU3 1/20 0.39
MAPK13 O15264 1/20 0.39
PTGS1 P23219 1/20 0.39
MAPK12 P53778 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22901548 0.91 MAPT (0.45) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901578 0.91 MAOB (0.48) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901555 0.91 MAOB (0.50) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901552 0.89 MAPT (0.43) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901547 0.89 MEN1 (0.51) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901563 0.85 MAOB (0.49) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901574 0.84 MAOB (0.47) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901607 0.83 MEN1 (0.38) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901571 0.82 MAPT (0.48) MAOBMEN1KMT2AMAPTHTT
SCHEMBL22901549 0.82 MAPT (0.48) MAOBMAPTHTTSMN1; SMN2GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021008588-A1 CLASS OF PYRIMIDINE QUINOLINE DERIVATIVES AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 广州新民培林医药科技有限公司 2021-01-21 WO disclosed