Laflunimus

Laflunimus

SCHEMBL22908

Cc1cc(NC(=O)/C(C#N)=C(\O)C2CC2)ccc1C(F)(F)F

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 6/20 0.67
LMNA P02545 1/20 0.39
KDR P35968 6/20 0.39
BRAF P15056 3/20 0.38
USP30 Q70CQ3 1/20 0.37
EPHX2 P34913 1/20 0.37
GAA P10253 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Laflunimus SCHEMBL9234178 1.00 DHODH (0.67) DHODHLMNAKDRBRAFUSP30
Laflunimus SCHEMBL21132 1.00 DHODH (0.67) DHODHLMNAKDRBRAFUSP30
Laflunimus SCHEMBL29677348 1.00 DHODH (0.67) DHODHLMNAKDRBRAFUSP30
SCHEMBL17100730 0.86 DHODH (0.49) DHODHKDRBRAFUSP30EPHX2
SCHEMBL21539519 0.86 DHODH (0.49) DHODHKDRBRAFUSP30EPHX2
SCHEMBL15196662 0.86 DHODH (0.62) DHODHLMNAGAATP53MAPT
SCHEMBL8717137 0.84 DHODH (0.66) DHODHLMNAGAATHRB
SCHEMBL8717143 0.84 DHODH (0.66) DHODHLMNAGAATHRB
SCHEMBL16274172 0.82 DHODH (0.58) DHODHGAATP53MAPTTHRB
SCHEMBL28236310 0.81 DHODH (0.49) DHODHLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 626 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4362968-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD47-SIRPA THERAPEUTIC AGENT Ohio State Innovation Foundation (US) 2024-05-08 EP claimed
US-20230303710-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD38 THERAPEUTIC AGENT OHIO STATE INNOVATION FOUNDATION (US) 2023-09-28 US claimed
WO-2023278778-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD47-SIRPΑ THERAPEUTIC AGENT OHIO STATE INNOVATION FOUNDATION (US) 2023-01-05 WO claimed
CN-115551488-A Nanoparticle compositions 艾格埃克斯制药有限公司 2022-12-30 CN claimed
EP-4081219-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD38 THERAPEUTIC AGENT Ohio State Innovation Foundation (US) 2022-11-02 EP claimed
WO-2021134045-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD38 THERAPEUTIC AGENT OHIO STATE INNOVATION FOUNDATION (US) 2021-07-01 WO claimed
EP-3829578-A1 SIROLIMUS CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2021-06-09 EP claimed
US-20200069661-A1 SIROLIMUS CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-03-05 US claimed
WO-2020047342-A1 SIROLIMUS CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-03-05 WO claimed
US-9668972-B2 Nonsteroidal immunomodulating kit and composition and uses thereof FOAMIX PHARMACEUTICALS LTD. (IL) 2017-06-06 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2008038147-A2 FOAMABLE VEHICLE COMPRISING DICARBOXYLIC ACID OR DICARBOXYLIC ACID ESTER AND PHARMACEUTICAL COMPOSITIONS THEREOF FOAMIX LTD. (US) 2008-04-03 WO claimed
US-20080044444-A1 Dicarboxylic acid foamable vehicle and pharmaceutical compositions thereof FOAMIX LTD. (IL) 2008-02-21 US claimed
EP-1863447-A2 NONSTEROIDAL IMMUNOMODULATING KIT AND COMPOSITION AND USES THEREOF Foamix Ltd. (IL) 2007-12-12 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
WO-2007007208-A2 NONSTEROIDAL IMMUNOMODULATING KIT AND COMPOSITION AND USES THEREOF FOAMIX LTD. (US) 2007-01-18 WO claimed
US-20060193789-A1 Surfacant, film forming agent, water, gas propellant; plant and animal extracts and oils; may include malathion FOAMIX LTD. (IL) 2006-08-31 US claimed
US-20050232869-A1 Nonsteroidal immunomodulating kit and composition and uses thereof FOAMIX LTD. 2005-10-20 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303710-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF DIHYDROOROTATE DEHYDROGENASE IN COMBINATION WITH AN ANTI-CD38 THERAPEUTIC AGENT DHODH, CD38, DPYD DHODH 1/4885LMNA 1972/4885KDR 3444/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.