SCHEMBL22909301

SCHEMBL22909301

O=C1CC(c2ccccc2Cl)=NN1c1ccc(Cl)cc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.62
MAPT P10636 6/20 0.62
MEN1 O00255 6/20 0.62
LMNA P02545 4/20 0.62
CD274 Q9NZQ7 5/20 0.60
PDCD1 Q15116 4/20 0.60
ALDH1A1 P00352 2/20 0.43
RAB9A P51151 1/20 0.43
GAA P10253 4/20 0.42
ALOX12 P18054 3/20 0.42
KDM4E B2RXH2 1/20 0.42
CASP6 P55212 2/20 0.41
TP53 P04637 2/20 0.41
CHRM2 P08172 1/20 0.39
ADRA2A P08913 1/20 0.39
OPRK1 P41145 1/20 0.39
PDE4D Q08499 1/20 0.39
MAOB P27338 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22909304 0.88 KMT2A (0.59) KMT2AMAPTMEN1LMNACD274
SCHEMBL22908672 0.85 PDCD1 (0.58) KMT2AMAPTMEN1LMNACD274
SCHEMBL10435326 0.85 MAPT (0.75) KMT2AMAPTMEN1LMNACD274
SCHEMBL22908674 0.82 KMT2A (0.70) KMT2AMAPTMEN1LMNACD274
SCHEMBL22909306 0.76 CYP3A4 (0.48) KMT2AMAPTMEN1LMNACD274
SCHEMBL11182553 0.76 PDCD1 (0.56) KMT2AMAPTMEN1LMNACD274
SCHEMBL10435333 0.76 MAPT (0.67) KMT2AMAPTMEN1LMNACD274
SCHEMBL22908687 0.75 CD274 (1.00) KMT2AMAPTMEN1LMNACD274
SCHEMBL17290401 0.75 CD274 (0.46) KMT2AMAPTMEN1LMNACD274
SCHEMBL22908646 0.74 KMT2A (0.61) KMT2AMAPTMEN1LMNACD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009384-A1 NOVEL PYRAZOLONE DERIVATIVES AS PD-1/PD-L1 INTERACTION INHIBITORS CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE LILLE (FR) 2021-01-21 WO disclosed