SCHEMBL22909304

SCHEMBL22909304

O=C1CC(c2ccccc2F)=NN1c1ccc(Cl)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.59
MAPT P10636 4/20 0.59
MEN1 O00255 3/20 0.59
LMNA P02545 2/20 0.59
CD274 Q9NZQ7 4/20 0.54
PDCD1 Q15116 3/20 0.54
MAOB P27338 3/20 0.45
CASP6 P55212 2/20 0.43
GAA P10253 2/20 0.43
HSD11B1 P28845 1/20 0.42
DRD3 P35462 2/20 0.41
OPRK1 P41145 2/20 0.41
HTR1A P08908 1/20 0.41
HTR3A P46098 1/20 0.41
KCNH2 Q12809 1/20 0.41
GHSR Q92847 1/20 0.41
ALDH1A1 P00352 1/20 0.39
ALOX12 P18054 1/20 0.39
KDM4E B2RXH2 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22909301 0.88 KMT2A (0.62) KMT2AMAPTMEN1LMNACD274
SCHEMBL22909306 0.88 CYP3A4 (0.48) KMT2AMAPTMEN1LMNACD274
SCHEMBL22908672 0.82 PDCD1 (0.58) KMT2AMAPTMEN1LMNACD274
SCHEMBL10435326 0.82 MAPT (0.75) KMT2AMAPTMEN1LMNACD274
SCHEMBL1661307 0.81 MEN1 (0.46) KMT2AMAPTMEN1CD274PDCD1
SCHEMBL22908674 0.79 KMT2A (0.70) KMT2AMAPTMEN1LMNACD274
SCHEMBL11895290 0.76 MEN1 (0.54) KMT2AMAPTMEN1CD274PDCD1
SCHEMBL11182553 0.73 PDCD1 (0.56) KMT2AMAPTMEN1LMNACD274
SCHEMBL10435333 0.73 MAPT (0.67) KMT2AMAPTMEN1LMNACD274
SCHEMBL10382658 0.72 MAOB (0.65) KMT2AMAPTMEN1LMNACD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009384-A1 NOVEL PYRAZOLONE DERIVATIVES AS PD-1/PD-L1 INTERACTION INHIBITORS CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE LILLE (FR) 2021-01-21 WO disclosed