SCHEMBL22918233

SCHEMBL22918233

Cc1occc1S(=O)(=O)C(F)(F)/C(F)=C/CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.35
ALDH1A1 P00352 4/20 0.32
TSHR P16473 2/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
HSD17B10 Q99714 2/20 0.31
CHRM2 P08172 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALOX15 P16050 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29486903 1.00 CASP3 (0.35) CASP3ALDH1A1TSHRMMP2MMP9
SCHEMBL28717560 0.84 CASP3 (0.38) CASP3ALDH1A1TSHRMMP2MMP9
SCHEMBL22918346 0.84 CASP3 (0.38) CASP3ALDH1A1TSHRMMP2MMP9
SCHEMBL29486893 0.84 CASP3 (0.38) CASP3ALDH1A1TSHRMMP2MMP9
SCHEMBL22918254 0.82 ALDH1A1 (0.42) CASP3ALDH1A1MMP2MMP9CA12
SCHEMBL22918257 0.81 CASP3 (0.39) CASP3TSHRMEN1KMT2ACA12
SCHEMBL29486875 0.81 CASP3 (0.39) CASP3TSHRMEN1KMT2ACA12
SCHEMBL22918282 0.80 CASP3 (0.42) CASP3ALDH1A1MMP2MMP9MEN1
SCHEMBL29486874 0.80 CASP3 (0.42) CASP3ALDH1A1MMP2MMP9MEN1
SCHEMBL28703648 0.80 CASP3 (0.42) CASP3ALDH1A1MMP2MMP9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114286816-A Difluoro-halogenated allylamine sulfone derivative inhibitor of lysyl oxidase, preparation method and application thereof 法玛西斯有限公司 2022-04-05 CN disclosed
WO-2021012014-A1 DIFLUOROHALOALLYLAMINE SULFONE DERIVATIVE INHIBITORS OF LYSYL OXIDASES, METHODS OF PREPARATION, AND USES THEREOF PHARMAXIS LTD. (AU) 2021-01-28 WO disclosed