SCHEMBL22919409

SCHEMBL22919409

COc1ccc(CNc2cc3cc(-c4ccccc4)c(-c4ccccc4)nc3cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 6/20 0.47
DYRK1A Q13627 2/20 0.47
MAPK13 O15264 1/20 0.47
RAF1 P04049 1/20 0.47
MAPK9 P45984 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
GAA P10253 2/20 0.47
HIF1A Q16665 2/20 0.46
TP53 P04637 3/20 0.46
MAPK1 P28482 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
TSHR P16473 2/20 0.46
CYP2C19 P33261 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ACP1 P24666 1/20 0.46
ALDH1A1 P00352 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31553220 1.00 CLK4 (0.47) CLK4DYRK1AMAPK13RAF1MAPK9
SCHEMBL22919333 0.78 PDGFRB (0.48) CLK4DYRK1AMAPK13RAF1MAPK9
SCHEMBL5223669 0.73 CLK4 (0.54) CLK4HIF1ATP53MAPK1CYP1A2
SCHEMBL27053625 0.73 CCNC (0.46) CLK4DYRK1AGAAHIF1ATP53
SCHEMBL27730117 0.72 HPGDS (0.54) CLK4DYRK1AGAAHIF1ATP53
SCHEMBL22919303 0.71 MAPT (0.51) GAAHIF1ATP53MAPK1HSD17B10
SCHEMBL20950754 0.69 CLK4 (0.50) CLK4DYRK1APTGDRMEN1KMT2A
SCHEMBL14330643 0.69 CLK4 (0.56) CLK4DYRK1AACP1KMT2AMAPT
SCHEMBL20489500 0.69 MAPT (0.57) CLK4DYRK1AGAALMNAMEN1
SCHEMBL2308761 0.68 NPC1 (0.68) CLK4DYRK1AGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269720-A acetyl-CoA synthetase short chains2(ACSS2) Small molecule inhibitors of 库拉德夫制药私人有限公司 2022-04-01 CN disclosed
WO-2021014415-A2 SMALL MOLECULE INHIBITORS OF ACETYL COENZYME A SYNTHETASE SHORT CHAIN 2 (ACSS2) CURADEV PHARMA PVT. LTD. (IN) 2021-01-28 WO disclosed