SCHEMBL22920182

SCHEMBL22920182

Fc1ccccc1NCc1ccc(C2CCCCC2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP1 O94782 1/20 0.42
WDR48 Q8TAF3 1/20 0.42
DGAT1 O75907 1/20 0.40
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
HTT P42858 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
GLA P06280 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP11B2 P19099 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAPK8 P45983 2/20 0.36
MAPK9 P45984 2/20 0.36
MAPK10 P53779 2/20 0.36
MAPK14 Q16539 2/20 0.36
CXCR4 P61073 1/20 0.36
PIM3 Q86V86 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22920035 0.81 MAOA (0.47) USP1WDR48KDM4EKMT2AL3MBTL1
SCHEMBL11511834 0.80 USP1 (0.48) USP1WDR48DGAT1KMT2AL3MBTL1
SCHEMBL22919961 0.79 HRH3 (0.44) KDM4EKMT2AL3MBTL1HTTTDP1
SCHEMBL22920027 0.78 NPC1 (0.41) KDM4EKMT2AL3MBTL1HTTTDP1
SCHEMBL20400977 0.77 STAT3 (0.52) KDM4EKMT2AL3MBTL1HTTTDP1
SCHEMBL20418716 0.75 USP1 (0.35) USP1WDR48KDM4EKMT2AL3MBTL1
SCHEMBL20401100 0.75 STAT3 (0.43) KMT2ATDP1SMN1; SMN2NPC1RAB9A
SCHEMBL20401141 0.75 STAT3 (0.42) USP1WDR48KDM4EKMT2AL3MBTL1
SCHEMBL29447666 0.74 USP1 (0.37) USP1WDR48KDM4EL3MBTL1NPC1
SCHEMBL20400421 0.74 STAT3 (0.41) KDM4EKMT2AL3MBTL1HTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021016333-A1 ARYL SULFONAMIDES AS SMALL MOLECULE STAT3 INHIBITORS UNIVERSITY OF HAWAII (US) 2021-01-28 WO disclosed