SCHEMBL22925792

SCHEMBL22925792

Cc1ccc(-c2cnc(Nc3ccc(C#N)nn3)o2)nc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.35
FLT1 P17948 3/20 0.35
FLT4 P35916 3/20 0.35
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
IMPDH2 P12268 3/20 0.32
GRM5 P41594 2/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 2/20 0.32
FAAH O00519 1/20 0.32
BPTF Q12830 1/20 0.32
EGLN2 Q96KS0 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
KEAP1 Q14145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22925604 0.86 KDR (0.35) KDRFLT1FLT4IMPDH2GRM5
SCHEMBL29620869 0.83 NPSR1 (0.39) KDRFLT1FLT4RAB9AKDM4E
SCHEMBL24636937 0.83 NPSR1 (0.39) KDRFLT1FLT4RAB9AKDM4E
SCHEMBL22925785 0.77 KDR (0.40) KDRFLT1FLT4CCR1CCR5
SCHEMBL22925712 0.76 ALOX5 (0.47) KDRFLT1FLT4IMPDH2RAB9A
SCHEMBL22925780 0.75 CCR1 (0.32) KDRFLT1FLT4CCR1CCR5
SCHEMBL22926082 0.73 TRPV1 (0.47) KDRFLT1FLT4IMPDH2
SCHEMBL29621019 0.73 KDR (0.39) KDRFLT1FLT4IMPDH2
SCHEMBL22925562 0.73 KDR (0.39) KDRFLT1FLT4IMPDH2
SCHEMBL22925966 0.70 CHEK1 (0.41) KDRFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021012018-A1 INHIBITOR COMPOUNDS Cincera Therapeutics Pty Ltd (AU) 2021-01-28 WO disclosed