SCHEMBL22925858

SCHEMBL22925858

COc1ccc(Oc2cc(C)ccc2N)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.60
ALDH1A1 P00352 6/20 0.55
CYP3A4 P08684 3/20 0.55
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
AR P10275 5/20 0.47
GAA P10253 1/20 0.46
BACE1 P56817 2/20 0.45
MEN1 O00255 2/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44
THRB P10828 1/20 0.44
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26394168 0.89 ALDH1A1 (0.61) ACHEALDH1A1CYP3A4CA12CA1
SCHEMBL22925860 0.83 ACHE (0.64) ACHEALDH1A1CYP3A4CA12CA1
SCHEMBL9517940 0.82 ALDH1A1 (0.66) ALDH1A1CYP3A4CA12CA1CA2
SCHEMBL10999189 0.82 TEAD4 (0.54) ACHEALDH1A1CYP3A4ARGAA
SCHEMBL12474539 0.82 ALDH1A1 (0.51) ALDH1A1CYP3A4CA12CA1CA2
SCHEMBL5583756 0.81 ALDH1A1 (0.63) ACHEALDH1A1CYP3A4ARGAA
SCHEMBL5583654 0.80 TEAD4 (0.57) ALDH1A1CYP3A4ARGAAMEN1
SCHEMBL22925857 0.80 ACHE (0.60) ACHEALDH1A1CYP3A4CA12CA1
SCHEMBL91459 0.80 ALDH1A1 (0.68) ACHEALDH1A1CYP3A4GAAMAPT
SCHEMBL30294328 0.80 ALDH1A1 (0.68) ACHEALDH1A1CYP3A4GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330477-B Phenyl thiophene sulfonamide compound, pharmaceutical composition, preparation method and application thereof 中国科学院上海有机化学研究所 2021-03-23 CN disclosed
WO-2021012689-A1 PHENYLTHIOPHENE SULFONAMIDE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海有机化学研究所 2021-01-28 WO disclosed
WO-2021012689-A1 PHENYLTHIOPHENE SULFONAMIDE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海有机化学研究所 2021-01-28 WO disclosed