SCHEMBL22932162

SCHEMBL22932162

O=C1CCC2(CCN(Cc3coc4ccccc34)C2)C(=O)N1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 9/20 0.60
DRD2 P14416 8/20 0.47
DRD4 P21917 8/20 0.47
DRD3 P35462 8/20 0.47
SIGMAR1 Q99720 2/20 0.45
HTR1A P08908 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21496463 0.77 CRBN (0.62) CRBNDRD2SIGMAR1ALDH1A1
SCHEMBL21496470 0.75 CRBN (1.00) CRBN
SCHEMBL22932163 0.74 DRD3 (0.50) CRBNDRD2DRD4DRD3HTR1A
SCHEMBL1750627 0.69 SIGMAR1 (0.58) DRD2DRD4DRD3SIGMAR1HTR1A
SCHEMBL22018722 0.69 CRBN (0.49) CRBN
SCHEMBL22932066 0.68 CRBN (0.50) CRBN
SCHEMBL28262836 0.67 ALDH1A1 (0.57) DRD2DRD4DRD3SIGMAR1HTR1A
SCHEMBL19586513 0.67 CRBN (0.55) CRBNALDH1A1
SCHEMBL22932089 0.66 CRBN (0.51) CRBN
SCHEMBL13772456 0.66 SIGMAR1 (0.58) DRD2DRD4DRD3SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11584748-B2 Spirocyclic compounds C4 THERAPEUTICS, INC. (US) 2023-02-21 US disclosed
US-20210032245-A1 SPIROCYCLIC COMPOUNDS C4 THERAPEUTICS, INC. (US) 2021-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210032245-A1 SPIROCYCLIC COMPOUNDS CRBN, RBX1, XIAP CRBN 1/4885DRD2 4192/4885DRD4 3894/4885
US-11584748-B2 Spirocyclic compounds CRBN, RBX1, XIAP CRBN 1/4885DRD2 4192/4885DRD4 3894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.