SCHEMBL22940384

SCHEMBL22940384

Cc1cccc2c1C(=O)N(C1CCC(=O)N(C)C1=O)C2=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 12/20 0.62
DDB1 Q16531 11/20 0.62
IKZF3 Q9UKT9 2/20 0.47
TNF P01375 1/20 0.47
IL1B P01584 1/20 0.47
TBXA2R P21731 1/20 0.47
IKZF1 Q13422 1/20 0.47
TMEM97 Q5BJF2 3/20 0.43
HTR2B P41595 2/20 0.43
ALDH1A1 P00352 1/20 0.40
CHRM2 P08172 1/20 0.40
OPRM1 P35372 1/20 0.40
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PDE6D O43924 1/20 0.40
STAT3 P40763 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9988681 0.90 DDB1 (0.60) CRBNDDB1IKZF3TNFIL1B
SCHEMBL19370936 0.89 CRBN (0.49) CRBNDDB1IKZF3TNFIL1B
SCHEMBL21062845 0.86 CRBN (0.60) CRBNDDB1IKZF3TNFIL1B
SCHEMBL21196697 0.86 DDB1 (0.60) CRBNDDB1IKZF3TNFIL1B
SCHEMBL32679446 0.86 CRBN (0.60) CRBNDDB1IKZF3TNFIL1B
SCHEMBL3797637 0.86 DDB1 (0.60) CRBNDDB1IKZF3TNFIL1B
SCHEMBL22649626 0.85 DDB1 (0.48) CRBNDDB1IKZF3TNFIL1B
SCHEMBL12041893 0.85 CRBN (0.53) CRBNDDB1IKZF3TNFIL1B
SCHEMBL845548 0.84 CRBN (0.54) CRBNDDB1IKZF3TNFIL1B
SCHEMBL24744448 0.84 DDB1 (0.49) CRBNDDB1IKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024108009-A1 DYRK/CLK PROTACS AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-05-23 WO disclosed
WO-2023249968-A1 BIFUNCTIONAL COMPOUNDS CONTAINING PYRIDO[2,3-DJPYRIMIDIN-7(8H)-ONE DERIVATIVES FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEASOME PATHWAY NIKANG THERAPEUTICS, INC. (US) 2023-12-28 WO disclosed
US-20230159559-A1 COMPOUND FOR INHIBITING AND INDUCING DEGRADATION OF EGFR KINASE BEIJING TIDE PHARMACEUTICAL CO., LTD. (CN) 2023-05-25 US disclosed
WO-2023088245-A1 DEGRADATION AGENT AND USE THEREOF 成都先导药物开发股份有限公司 2023-05-25 WO disclosed
WO-2022068849-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADATION OF EGFR AND RELATED METHODS OF USE BEIGENE, LTD. (KY) 2022-04-07 WO disclosed
WO-2021018018-A1 DEGRADATION OF BRUTON'S TYROSINE KINASE (BTK) BY CONJUGATION OF BTK INIDBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE BEIGENE, LTD. (KY) 2021-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159559-A1 COMPOUND FOR INHIBITING AND INDUCING DEGRADATION OF EGFR KINASE EGFR, ERBB2, ERBB3 CRBN 898/4885DDB1 2765/4885IKZF3 1670/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.