SCHEMBL22944210

SCHEMBL22944210

CN1CCC(COc2cc(Nc3cnc(C#N)cn3)nnc2I)CC1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 20/20 0.55
CHEK2 O96017 2/20 0.48
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22944207 0.88 CHEK1 (0.55) CHEK1CHEK2
SCHEMBL22944214 0.87 CHEK1 (0.57) CHEK1CHEK2KCNH2
SCHEMBL22943220 0.77 CHEK1 (0.68) CHEK1CHEK2
SCHEMBL22943209 0.76 CHEK1 (0.65) CHEK1CHEK2
SCHEMBL22944206 0.76 CHEK1 (0.56) CHEK1CHEK2KCNH2
SCHEMBL22944582 0.75 CHEK1 (0.64) CHEK1CHEK2KCNH2
SCHEMBL22944600 0.75 CHEK1 (0.64) CHEK1CHEK2
SCHEMBL22943424 0.75 CHEK1 (0.64) CHEK1CHEK2
SCHEMBL22943232 0.75 CHEK1 (0.61) CHEK1CHEK2
SCHEMBL22943190 0.74 CHEK1 (0.62) CHEK1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021019514-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITOR AND USES THEREOF INTEGRAL BIOSCIENCES PVT. LTD. (IN) 2021-02-04 WO disclosed