SCHEMBL22959236

SCHEMBL22959236

COc1ncc(Oc2c(Cl)ccc(N)c2Cl)cc1C(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 9/20 0.47
P2RX3 P56373 3/20 0.36
P2RX2 Q9UBL9 3/20 0.36
THRB P10828 2/20 0.36
MAPT P10636 1/20 0.35
CASP1 P29466 1/20 0.35
AURKA O14965 1/20 0.35
TTK P33981 1/20 0.35
AURKB Q96GD4 1/20 0.35
INCENP Q9NQS7 1/20 0.35
PDCD1 Q15116 2/20 0.34
CD274 Q9NZQ7 2/20 0.34
NPBWR1 P48145 2/20 0.34
MCHR1 Q99705 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22959108 0.82 RORC (0.47) RORCP2RX3P2RX2THRBNPBWR1
SCHEMBL29527631 0.82 RORC (0.53) RORCP2RX3P2RX2THRBMAPT
SCHEMBL22959151 0.82 RORC (0.53) RORCP2RX3P2RX2THRBMAPT
SCHEMBL22959254 0.81 RORC (0.51) RORCP2RX3P2RX2THRB
SCHEMBL29872245 0.81 RORC (0.51) RORCP2RX3P2RX2THRB
SCHEMBL24449964 0.77 RORC (0.46) RORCP2RX3P2RX2THRBMAPT
SCHEMBL24449957 0.77 RORC (0.43) RORCP2RX3P2RX2THRBMAPT
SCHEMBL24449959 0.76 RORC (0.41) RORCP2RX3P2RX2THRBMAPT
SCHEMBL30558158 0.76 RORC (0.41) RORCP2RX3P2RX2THRBMAPT
SCHEMBL22959061 0.75 RORC (0.51) RORCTHRBMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021026179-A1 AGONISTS OF ROR GAMMAt BRISTOL-MYERS SQUIBB COMPANY (US) 2021-02-11 WO disclosed