SCHEMBL2298402

SCHEMBL2298402

C[O+]=C(N(C)C)N(C)n1nnc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 9/20 0.42
POLB P06746 2/20 0.42
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
KEAP1 Q14145 1/20 0.42
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DGAT1 O75907 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
THPO P40225 1/20 0.39
CYP4Z1 Q86W10 1/20 0.39
KCNMA1 Q12791 2/20 0.36
MGAM O43451 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3919726 0.94 SLC9A1 (0.38) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL5713206 0.78 FAAH (0.37)
SCHEMBL4958142 0.75 NPSR1 (0.42) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL31130802 0.75 SLC9A1 (0.55) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL28863784 0.75 SLC9A1 (0.55) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL30378712 0.73 SLC9A1 (0.46) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL78773 0.73 SLC9A1 (0.46) SLC9A1POLBMAPK1ATMKEAP1
Bromide SCHEMBL5514455 0.72 SLC9A1 (0.44) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL1462681 0.72 SLC9A1 (0.44) SLC9A1POLBMAPK1ATMKEAP1
SCHEMBL5090298 0.72 SLC9A1 (0.44) SLC9A1POLBMAPK1ATMKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263800-B1 LINKER BASED SOLID SUPPORT FOR PEPTIDE AND SMALL MOLECULE ORGANIC SYNTHESIS COUNCIL SCIENT IND RES (IN) 2006-11-08 EP claimed
US-7994118-B2 Template fixed beta-hairpin loop mimetics and their use in phage display POLYPHOR LTD. (CH) 2011-08-09 US disclosed
WO-1992019254-A1 α-SUBSTITUTED POLYPEPTIDES HAVING THERAPEUTIC ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-11-12 WO disclosed