SCHEMBL22988124

SCHEMBL22988124

C[S+]([O-])c1cccc(-c2nc3c4ccccc4nc(N)n3n2)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.48
ADORA1 P30542 3/20 0.48
ADORA2A P29274 1/20 0.47
RXFP1 Q9HBX9 1/20 0.44
TP53 P04637 1/20 0.44
THRB P10828 1/20 0.42
MAPT P10636 3/20 0.42
POLB P06746 1/20 0.42
PDPK1 O15530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22987825 0.80 CSNK1D (0.59) ADORA3ADORA1ADORA2ARXFP1TP53
SCHEMBL22987873 0.79 ADORA3 (0.50) ADORA3ADORA1ADORA2ARXFP1TP53
SCHEMBL22988327 0.74 ADORA1 (0.47) ADORA3ADORA1ADORA2ARXFP1TP53
SCHEMBL743593 0.73 RXFP1 (0.58) ADORA3ADORA1ADORA2ARXFP1TP53
SCHEMBL22988309 0.72 ADORA3 (0.53) ADORA3ADORA1ADORA2ATP53MAPT
SCHEMBL22988304 0.72 ADORA3 (0.65) ADORA3ADORA1ADORA2ATHRBMAPT
SCHEMBL22988235 0.71 ADORA3 (0.51) ADORA3ADORA1ADORA2ATP53MAPT
SCHEMBL22988361 0.70 PDE10A (0.53) ADORA3ADORA1ADORA2ARXFP1THRB
SCHEMBL18948427 0.69 PDE10A (0.63) ADORA3ADORA1TP53PDPK1
SCHEMBL24209870 0.68 ADORA3 (0.71) ADORA3ADORA1ADORA2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed