SCHEMBL23015341

SCHEMBL23015341

C#Cc1cc(N)c(C(=O)OC)cc1F

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 6/20 0.49
CFTR P13569 7/20 0.46
GAA P10253 5/20 0.45
HSD17B10 Q99714 3/20 0.45
HPGD P15428 3/20 0.45
MAPT P10636 2/20 0.45
GLA P06280 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
ATM Q13315 1/20 0.45
ABL1 P00519 1/20 0.44
TSHR P16473 2/20 0.43
ALOX15 P16050 1/20 0.43
POLB P06746 1/20 0.40
IKBKB O14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL195591 0.81 KDM4E (0.61) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL2900514 0.80 KDM4E (0.59) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL23015343 0.80 KDM4E (0.51) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL12021817 0.79 KDM4E (0.51) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL24324843 0.78 KDM4E (0.58) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL29611549 0.78 KDM4E (0.58) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL16411016 0.78 KDM4E (0.50) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL2391637 0.78 CFTR (0.63) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL24413980 0.77 KDM4E (0.47) KDM4EALDH1A1CFTRGAAHSD17B10
SCHEMBL3616519 0.77 KDM4E (0.56) KDM4EALDH1A1CFTRGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4017593-B1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING SCRIPPS RESEARCH INST (US) 2025-07-23 EP disclosed
CN-115003383-B Bicyclic agonists of the interferon Gene stimulator STING 斯克里普斯研究学院 2024-10-01 CN disclosed
US-20220332720-A1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING THE SCRIPPS RESEARCH INSTITUTE 2022-10-20 US disclosed
CN-115003383-A Bicyclic agonists of interferon gene stimulator STING 斯克里普斯研究学院 2022-09-02 CN disclosed
EP-4017593-A1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING The Scripps Research Institute (US) 2022-06-29 EP disclosed
WO-2021035258-A1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING THE SCRIPPS RESEARCH INSTITUTE (US) 2021-02-25 WO disclosed
WO-2021035258-A1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING THE SCRIPPS RESEARCH INSTITUTE (US) 2021-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220332720-A1 BICYCLIC AGONISTS OF STIMULATOR OF INTERFERON GENES STING STING1, IRF3, IFNAR1 KDM4E 1800/4885ALDH1A1 3495/4885CFTR 641/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.