SCHEMBL23020137

SCHEMBL23020137

N#Cc1cc(-c2ccc(-c3ccccn3)cc2)cc(-c2ccc(-c3ccc(-c4nc(-c5ccccc5)nc(-c5ccccc5)n4)cc3)c3ccccc23)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 9/20 0.49
ABCG2 Q9UNQ0 4/20 0.40
SQOR Q9Y6N5 1/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
MAPK1 P28482 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
TGFBR1 P36897 1/20 0.39
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23020076 0.95 GRM5 (0.47) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL23020430 0.95 GRM5 (0.52) GRM5ABCG2SQORTSHRHSD17B10
SCHEMBL23020170 0.92 GRM5 (0.56) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL23020162 0.91 MEN1 (0.44) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL23020186 0.90 GRM5 (0.55) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL23020185 0.90 GRM5 (0.55) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL21098948 0.90 TSHR (0.46) TSHRHSD17B10MAPK1MEN1ALDH1A1
SCHEMBL23020309 0.89 GRM5 (0.44) GRM5ABCG2TSHRHSD17B10CLK4
SCHEMBL22652775 0.89 MAPK1 (0.48) GRM5ABCG2TSHRHSD17B10MAPK1
SCHEMBL23020172 0.88 GRM5 (0.49) GRM5SQORTGFBR1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3392242-B1 NOVEL HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME LG CHEMICAL LTD (KR) 2021-02-24 EP disclosed