SCHEMBL23020430

SCHEMBL23020430

N#Cc1cc(-c2ccccn2)cc(-c2ccc(-c3ccc(-c4nc(-c5ccccc5)nc(-c5ccccc5)n4)cc3)c3ccccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 9/20 0.52
ABCG2 Q9UNQ0 3/20 0.42
SQOR Q9Y6N5 1/20 0.41
CLK4 Q9HAZ1 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNH2 Q12809 1/20 0.41
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23020137 0.95 GRM5 (0.49) GRM5ABCG2SQORCLK4MEN1
SCHEMBL23020076 0.91 GRM5 (0.47) GRM5ABCG2CLK4MEN1ALDH1A1
SCHEMBL21099056 0.90 KDM4E (0.46) MEN1ALDH1A1LMNATSHRKMT2A
SCHEMBL21099059 0.88 SMN1; SMN2 (0.46) MEN1ALDH1A1LMNATSHRKMT2A
SCHEMBL23020162 0.88 MEN1 (0.44) GRM5ABCG2CLK4MEN1ALDH1A1
SCHEMBL19939360 0.87 CYP1A2 (0.50) ABCG2CLK4MEN1ALDH1A1LMNA
SCHEMBL23020170 0.86 GRM5 (0.56) GRM5ABCG2CLK4MEN1ALDH1A1
SCHEMBL20195361 0.86 KDM4E (0.44) GRM5MEN1ALDH1A1LMNATSHR
SCHEMBL23020309 0.85 GRM5 (0.44) GRM5ABCG2CLK4MEN1ALDH1A1
SCHEMBL23020186 0.85 GRM5 (0.55) GRM5ABCG2CLK4MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3392242-B1 NOVEL HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME LG CHEMICAL LTD (KR) 2021-02-24 EP disclosed