SCHEMBL23022320

SCHEMBL23022320

OCc1ccc2nn(I)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.37
CA2 P00918 3/20 0.34
CA12 O43570 2/20 0.34
CA3 P07451 2/20 0.34
CA4 P22748 2/20 0.34
CA6 P23280 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
CA5B Q9Y2D0 2/20 0.34
CA5A P35218 1/20 0.34
APP P05067 2/20 0.33
CBFB Q13951 2/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
ESR2 Q92731 1/20 0.33
RPS6KA5 O75582 1/20 0.32
RECQL P46063 1/20 0.32
TYR P14679 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3436381 0.79 KDM4E (0.49) HSD17B10CA2CA12CA3CA4
SCHEMBL904586 0.76 SLC5A2 (0.46) HSD17B10APPRPS6KA5HDAC6
SCHEMBL15971092 0.75 SLC5A2 (0.47) HSD17B10CA2CA12CA3CA4
SCHEMBL15687224 0.72 HDAC6 (0.45) ESR2HDAC6
SCHEMBL19763377 0.71 ESR2 (0.47) HSD17B10ESR2
SCHEMBL15687365 0.69 ALDH1A1 (0.36) HSD17B10CBFBHDAC6
SCHEMBL21575908 0.68 NPC1 (0.40) HSD17B10TYRPDE10A
SCHEMBL16152984 0.68 CYP1A2 (0.41) HSD17B10
SCHEMBL1206769 0.66 CA2 (0.54) HSD17B10CA2CA12CA3CA4
SCHEMBL29749150 0.66 CA2 (0.54) HSD17B10CA2CA12CA3CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021032148-A1 AMINOPYRAZINE COMPOUNDS AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2021-02-25 WO disclosed