SCHEMBL230242

SCHEMBL230242

O=C(O)C(O)C(ON1C(=O)CCC1=O)(C(=O)O)N1C(=O)CCC1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16875685 0.72 CA12 (0.32)
SCHEMBL23781544 0.70 CPT2 (0.34)
SCHEMBL2570752 0.70
SCHEMBL16875690 0.70
SCHEMBL57128 0.62 PARL (0.38)
SCHEMBL1350795 0.62 PARL (0.31)
SCHEMBL1350799 0.62 PARL (0.31)
SCHEMBL230241 0.61 PARL (0.34)
SCHEMBL379296 0.61 PARL (0.34)
SCHEMBL16875684 0.61 MGLL (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 490 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2971064-B1 PROXIMITY ASSAY FOR IN SITU DETECTION OF TARGETS VENTANA MED SYST INC (US) 2019-10-16 EP claimed
US-9663814-B2 Proximity assay for in situ detection of targets VENTANA MEDICAL SYSTEMS, INC. (US) 2017-05-30 US claimed
EP-1853634-B1 ACTIVATED SIALIC ACID DERIVATIVES FOR PROTEIN DERIVATISATION AND CONJUGATION LIPOXEN TECHNOLOGIES LTD (GB) 2016-08-10 EP claimed
EP-2971064-A1 PROXIMITY ASSAY FOR IN SITU DETECTION OF TARGETS Ventana Medical Systems, Inc. (US) 2016-01-20 EP claimed
US-20160002701-A1 Proximity Assay for In Situ Detection of Targets VENTANA MEDICAL SYSTEMS, INC. 2016-01-07 US claimed
WO-2014139980-A1 PROXIMITY ASSAY FOR IN SITU DETECTION OF TARGETS VENTANA MEDICAL SYSTEMS, INC. (US) 2014-09-18 WO claimed
WO-2014139979-A1 QUANTUM DOT IN SITU HYBRIDIZATION VENTANA MEDICAL SYSTEMS, INC. (US) 2014-09-18 WO claimed
EP-2276499-B1 RECOMBINANT DEAMIDATED GLIADIN ANTIGEN BIO RAD LABORATORIES (US) 2013-06-12 EP claimed
US-5427929-A Enzyme pretreatment AMGEN INC. (US) 1995-06-27 US claimed
WO-1988008875-A1 CYCLING BIOCHIP SENSOR THE WASHINGTON TECHNOLOGY CENTER (US) 1988-11-17 WO claimed
EP-4743220-A1 DRIED REAGENTS Olink Proteomics AB (SE) 2026-05-20 EP disclosed
EP-4743076-A2 SYNTHETIC BI-FUNCTIONAL DEGRADERS OF INTEGRINS The Board of Trustees of the Leland Stanford Junior University (US) 2026-05-20 EP disclosed
EP-3600372-B1 SYNTHEKINE COMPOSITIONS AND METHODS OF USE UNIV LELAND STANFORD JUNIOR (US) 2026-05-13 EP disclosed
US-12601683-B2 Serial multichannel microscopy Miltenyi Biotec B.V. & Co. KG (DE) 2026-04-14 US disclosed
EP-4441079-B1 SWITCHABLE POLYPEPTIDE AND ITS USE FOR GENTLE AFFINITY PURIFICATION UNIV OXFORD INNOVATION LTD (GB) 2026-02-11 EP disclosed
EP-0481069-A1 METHOD FOR REDUCING CARRYOVER CONTAMINATION IN AN AMPLIFICATION PROCEDURE AMGEN INC. (US) 1992-04-22 EP disclosed
US-5094950-A Diagnostics NIHON MEDI-PHYSICS CO., LTD. (JP) 1992-03-10 US disclosed
WO-1991017270-A1 METHOD FOR REDUCING CARRYOVER CONTAMINATION IN AN AMPLIFICATION PROCEDURE AMGEN INC. (US) 1991-11-14 WO disclosed
EP-0345723-A2 Diethylenetriamine pentaacetic acid derivatives NIHON MEDI-PHYSICS CO., LTD. (JP) 1989-12-13 EP disclosed
WO-1988008875-A1 CYCLING BIOCHIP SENSOR THE WASHINGTON TECHNOLOGY CENTER (US) 1988-11-17 WO disclosed