SCHEMBL23029979

SCHEMBL23029979

Cc1nc2c(Br)ccc(Cl)n2n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 6/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
PDE10A Q9Y233 6/20 0.35
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
TP53 P04637 1/20 0.33
AHR P35869 1/20 0.33
PDE5A O76074 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE4A P27815 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23029946 0.81 HAVCR2 (0.39) HAVCR2HPGDLMNATSHRPDE10A
SCHEMBL23029977 0.75 HAVCR2 (0.35) HAVCR2HPGDLMNATSHRPDE10A
SCHEMBL16565475 0.65 AHR (0.54) HAVCR2HPGDPDE10AHSD17B10MAPT
SCHEMBL19761029 0.65 LMNA (0.38) HAVCR2HPGDLMNATSHRPDE10A
SCHEMBL1044937 0.65 CHEK1 (0.34)
SCHEMBL405895 0.63 PDE10A (0.57) HAVCR2PDE10APDE5APDE4D
SCHEMBL31167556 0.63 PDE10A (0.57) HAVCR2LMNAPDE10AHSD17B10MAPT
SCHEMBL25342261 0.62 KDM4E (0.35) HAVCR2HPGDLMNAPDE10AL3MBTL1
SCHEMBL19761037 0.62 TLR9 (0.34) L3MBTL1MAPT
SCHEMBL31329841 0.62 HAVCR2 (0.36) HAVCR2HPGDLMNATSHRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4019521-A1 AZAHETEROARYL COMPOUND AND APPLICATION THEREOF Blueray Therapeutics (Shanghai) Co., Ltd (CN) 2022-06-29 EP disclosed
WO-2021032004-A9 AZAHETEROARYL COMPOUND AND APPLICATION THEREOF 上海青煜医药科技有限公司 2021-03-25 WO disclosed
WO-2021032004-A1 AZAHETEROARYL COMPOUND AND APPLICATION THEREOF 上海青煜医药科技有限公司 2021-02-25 WO disclosed