SCHEMBL2304116

SCHEMBL2304116

CCCCN(C(=O)O)C1CCC(C)NC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
ADH1C P00326 1/20 0.32
ADH1A P07327 1/20 0.32
ADH4 P08319 1/20 0.32
SLC6A2 P23975 7/20 0.32
SLC6A4 P31645 7/20 0.32
SLC6A3 Q01959 4/20 0.31
KCNH2 Q12809 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
PTBP1 P26599 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3821799 0.80 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL1221462 0.80 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL28246290 0.80 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL2875169 0.77 SLC6A2 (0.41) L3MBTL1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL17786300 0.77 SLC6A2 (0.41) L3MBTL1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL1932588 0.76 L3MBTL1 (0.41) L3MBTL1ADH1CADH1AADH4CYP3A4
SCHEMBL3818321 0.76 SLC6A4 (0.44) SIGMAR1L3MBTL1SLC6A2SLC6A4SLC6A3
SCHEMBL18704813 0.75 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL13736459 0.74 L3MBTL1 (0.35) SIGMAR1L3MBTL1SLC6A2SLC6A4CYP3A4
SCHEMBL5510945 0.74 L3MBTL1 (0.42) L3MBTL1ADH1CADH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349269-A1 2,5-DISUBSTITUTED PIPERIDINE OREXIN RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-08-03 EP disclosed
WO-2010048012-A1 2,5-DISUBSTITUTED PIPERIDINE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-04-29 WO disclosed