SCHEMBL23043365

SCHEMBL23043365

CC(C)(C)OC(=O)N1C2CCC1(C(N)=O)CN(C(c1ccccc1)(c1ccccc1)c1ccccc1)C2

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.35
RORC P51449 11/20 0.35
KDM1A O60341 1/20 0.35
HDAC1 Q13547 1/20 0.33
USP30 Q70CQ3 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
HSD11B1 P28845 1/20 0.33
CCR5 P51681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23043737 0.92 GPR119 (0.37) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL30962981 0.89 GPR119 (0.35) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL23053525 0.89 GPR119 (0.35) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL23042967 0.84 RORC (0.39) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL30759505 0.83 RORC (0.38) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL31386491 0.83 RORC (0.38) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL30759653 0.83 RORC (0.38) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL23042964 0.83 GPR119 (0.37) GPR119RORCKDM1AUSP30KDM4E
SCHEMBL30089167 0.82 KDM1A (0.36) GPR119RORCKDM1AKDM4EPKM
SCHEMBL25244104 0.82 ABCB1 (0.39) GPR119RORCKDM1AKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114615981-B KRAS G12D inhibitors 米拉蒂治疗股份有限公司 2024-04-12 CN disclosed
US-20230279025-A1 KRAS G12D INHIBITORS ARRAY BIOPHARMA INC. 2023-09-07 US disclosed
US-20230279025-A1 KRAS G12D INHIBITORS ARRAY BIOPHARMA INC. 2023-09-07 US disclosed
EP-4021444-A1 KRAS G12D INHIBITORS Mirati Therapeutics, Inc. (US) 2022-07-06 EP disclosed
CN-114615981-A KRAS G12D inhibitors 米拉蒂治疗股份有限公司 2022-06-10 CN disclosed
WO-2021041671-A1 KRAS G12D INHIBITORS Mirati Therapeutics, Inc. (US) 2021-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230279025-A1 KRAS G12D INHIBITORS KRAS, NRAS, HRAS GPR119 1751/4885RORC 874/4885KDM1A 3361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.