SCHEMBL23048780

SCHEMBL23048780

Fc1cc(OCc2ccccc2)c(-n2cc(C3CC3)nc2S)cc1Br

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.37
HTR1A P08908 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
PTGER1 P34995 1/20 0.34
S1PR5 Q9H228 1/20 0.33
PRMT5 O14744 3/20 0.33
IDO1 P14902 1/20 0.33
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23048781 0.82 MAP3K5 (0.39) KDM1AHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL23865458 0.82 MAP3K5 (0.36) SLC6A4
SCHEMBL23865352 0.81 HCRTR1 (0.30)
SCHEMBL30809618 0.73 SLC6A4 (0.48) KDM1AHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL27090021 0.73 SLC6A4 (0.48) KDM1AHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL23048746 0.72 MAP3K5 (0.31)
SCHEMBL23048795 0.72 RAB9A (0.36)
SCHEMBL23048617 0.70
SCHEMBL416139 0.68 KDM1A (0.48) KDM1AHTR1APTGER1S1PR5
SCHEMBL22473952 0.68 MAP3K5 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3572401-B1 ASK1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF FUJIAN COSUNTER PHARMACEUTICAL CO LTD (CN) 2021-09-29 EP disclosed
EP-3572412-B1 PYRIDINE DERIVATIVE AS ASK1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF FUJIAN COSUNTER PHARMACEUTICAL CO LTD (CN) 2021-03-03 EP disclosed