SCHEMBL23058729

SCHEMBL23058729

CCCN(C(C)C)C(C)c1ccc(OC(F)(F)F)cc1F

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 9/20 0.52
GPR139 Q6DWJ6 3/20 0.41
IDH1 O75874 3/20 0.35
HDAC6 Q9UBN7 1/20 0.34
GPR3 P46089 2/20 0.34
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23058771 0.80 MC4R (0.39) HDAC6
SCHEMBL23058487 0.79 PDE2A (0.47) PDE2AHDAC6
SCHEMBL12883103 0.75 PDE2A (0.63) PDE2AGPR139IDH1GPR3
SCHEMBL23059051 0.74 PDE2A (0.48) PDE2A
SCHEMBL18290665 0.72 PDE2A (0.60) PDE2AGPR139IDH1GPR3
SCHEMBL16043293 0.72 PDE2A (0.60) PDE2AGPR139GPR3
SCHEMBL30557811 0.72 PDE2A (0.60) PDE2AGPR139GPR3
SCHEMBL17769060 0.72 PDE2A (0.60) PDE2AGPR139GPR3
SCHEMBL23058728 0.71 PDE2A (0.44) PDE2ANR1H2NR1H3
SCHEMBL23058734 0.71 PDE2A (0.44) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021041588-A1 SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-03-04 WO disclosed