SCHEMBL23058728

SCHEMBL23058728

CCCCN(C(C)C)C(C)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.44
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
ALDH1A1 P00352 2/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
SLC7A5 Q01650 2/20 0.36
EPHX1 P07099 1/20 0.36
PPARG P37231 2/20 0.36
PPARD Q03181 2/20 0.36
PPARA Q07869 2/20 0.36
CRHR1 P34998 1/20 0.35
TSHR P16473 1/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
CYP2C9 P11712 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23058487 0.91 PDE2A (0.47) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL23058734 0.77 PDE2A (0.44) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL20746964 0.75 PDE2A (0.47) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL19506428 0.75 PDE2A (0.48) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL28183071 0.74 HDAC3 (0.47) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL19506041 0.74 PDE2A (0.46) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL2093549 0.73 PDE2A (0.53) PDE2AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL10087166 0.73 PDE2A (0.49) PDE2AALDH1A1SLC7A5SLC6A4SLC6A3
SCHEMBL10087250 0.73 PDE2A (0.51) PDE2AALDH1A1SLC7A5EPHX1SLC6A4
SCHEMBL1728974 0.73 SLC2A1 (0.55) PDE2AHDAC3HDAC1HDAC2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021041588-A1 SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-03-04 WO disclosed