SCHEMBL23058734

SCHEMBL23058734

CCCN(C(C)C)C(CC)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.44
ALDH1A1 P00352 2/20 0.38
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
EPHX1 P07099 1/20 0.36
TSHR P16473 1/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
HRH3 Q9Y5N1 2/20 0.34
CRHR1 P34998 2/20 0.34
SLC7A5 Q01650 2/20 0.34
LMNA P02545 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23058487 0.85 PDE2A (0.47) PDE2AALDH1A1EPHX1TSHRSLC6A4
SCHEMBL23058728 0.77 PDE2A (0.44) PDE2AALDH1A1EPHX1TSHRSLC6A4
SCHEMBL12318715 0.73 PDE2A (0.56) PDE2AALDH1A1EPHX1TSHRSLC6A4
SCHEMBL14233628 0.73 PDE2A (0.56) PDE2AALDH1A1EPHX1TSHRSLC6A4
SCHEMBL23058729 0.71 PDE2A (0.52) PDE2A
SCHEMBL20032388 0.71 PDE2A (0.53) PDE2AALDH1A1TSHRHRH3LMNA
SCHEMBL17914547 0.71 TSHR (0.46) PDE2AALDH1A1EPHX1TSHRSLC6A4
SCHEMBL23058782 0.71 NPSR1 (0.36) ALDH1A1SLC7A5
SCHEMBL23058137 0.71 CRHR1 (0.40) PDE2ATSHRSLC6A4HRH3CRHR1
SCHEMBL20381850 0.70 PDE2A (0.53) PDE2AALDH1A1EPHX1TSHRSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021041588-A1 SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-03-04 WO disclosed