SCHEMBL23060201

SCHEMBL23060201

C=CC(=O)Nc1cc(OC(F)(F)F)ccc1C(=O)OCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTO1 P78417 1/20 0.47
TP53 P04637 1/20 0.46
LMNA P02545 1/20 0.45
ALDH1A1 P00352 3/20 0.44
POLB P06746 2/20 0.43
JAK3 P52333 5/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.43
THRB P10828 1/20 0.43
TEAD1 P28347 1/20 0.42
MCL1 Q07820 1/20 0.41
FGFR4 P22455 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
TEK Q02763 1/20 0.40
CDC25B P30305 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23044925 0.88 ALDH1A1 (0.46) ALDH1A1POLBSMN1; SMN2GAATHRB
SCHEMBL23044920 0.87 GSTO1 (0.44) GSTO1LMNAALDH1A1JAK3SMN1; SMN2
SCHEMBL21430983 0.86 ALDH1A1 (0.50) GSTO1TP53LMNAALDH1A1JAK3
SCHEMBL23044908 0.85 GSTO1 (0.43) GSTO1TP53LMNAALDH1A1JAK3
SCHEMBL29214307 0.84 GSTO1 (0.45) GSTO1LMNAALDH1A1JAK3SMN1; SMN2
SCHEMBL21430738 0.81 GSTO1 (0.45) GSTO1LMNAALDH1A1POLBJAK3
Hydrochloric Acid SCHEMBL3962928 0.81 POLB (0.48) TP53LMNAALDH1A1POLBSMN1; SMN2
SCHEMBL29214310 0.81 GSTO1 (0.43) GSTO1TP53LMNAALDH1A1POLB
SCHEMBL21332113 0.81 TP53 (0.46) TP53LMNAALDH1A1POLBSMN1; SMN2
SCHEMBL21430909 0.80 HPGD (0.47) GSTO1LMNAALDH1A1JAK3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4023639-A1 PYRAZOLE DERIVATIVE FOR FGFR INHIBITOR AND PREPARATION METHOD THEREFOR Etern Biopharma (Shanghai) Co., Ltd. (CN) 2022-07-06 EP disclosed
WO-2021037219-A1 PYRAZOLE DERIVATIVE FOR FGFR INHIBITOR AND PREPARATION METHOD THEREFOR 上海奕拓医药科技有限责任公司 2021-03-04 WO disclosed