SCHEMBL2306499

SCHEMBL2306499

FC(F)(F)Oc1cccc(Br)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.43
IDH1 O75874 3/20 0.38
IDH2 P48735 1/20 0.38
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA3 P34903 1/20 0.32
SCN5A Q14524 1/20 0.31
MPL P40238 1/20 0.31
TGFBR1 P36897 1/20 0.30
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31445247 1.00 HTR7 (0.43) HTR7IDH1IDH2GABRA1GABRG2
SCHEMBL4452048 0.79 HTR7 (0.47) HTR7HTR1ADRD2
SCHEMBL2302960 0.75 CYP3A4 (0.42) IDH1IDH2MPL
SCHEMBL30319918 0.75 NOS3 (0.40) IDH1IDH2SCN5AMPL
SCHEMBL20049307 0.75 IDH1 (0.38) IDH1IDH2MPLTGFBR1HTR1A
SCHEMBL16289639 0.75 IDH1 (0.38) IDH1IDH2MPLTGFBR1HTR1A
SCHEMBL2302655 0.75 NOS3 (0.40) IDH1IDH2SCN5AMPL
SCHEMBL13680498 0.75 CCR1 (0.43) IDH1IDH2GRM5
SCHEMBL3386747 0.75 HTR7 (0.51) HTR7GABRA1GABRG2GABRB3GABRA3
SCHEMBL22489576 0.75 IDH1 (0.39) IDH1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350008-B1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2012-09-05 EP disclosed
EP-2350008-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES Bayer CropScience AG (DE) 2011-08-03 EP disclosed
WO-2010040461-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2010-04-15 WO disclosed