SCHEMBL2306989

SCHEMBL2306989

Cc1c(C(=O)O)c2c([C@@H](c3cc(F)cc(F)c3C(N)=O)C3CCC3)ccc(F)c2c(=O)n1Cc1ncco1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 5/20 0.35
MDM2 Q00987 14/20 0.34
TP53 P04637 1/20 0.31
GLP1R P43220 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2313391 0.91 S1PR3 (0.34) S1PR3MDM2GLP1R
SCHEMBL3345533 0.88 S1PR3 (0.36) S1PR3
SCHEMBL2308354 0.88 S1PR3 (0.33) S1PR3GLP1R
SCHEMBL2306426 0.81 CYP2C9 (0.35) S1PR3
SCHEMBL2356247 0.75 MAPT (0.31) MDM2
SCHEMBL2311690 0.74 GNRHR (0.35)
SCHEMBL2310282 0.74 FEN1 (0.38) S1PR3GLP1R
SCHEMBL2313425 0.72 GNRHR (0.39) S1PR3MDM2
SCHEMBL1364329 0.70 S1PR3 (0.38) S1PR3
SCHEMBL1367105 0.69 CYP1B1 (0.39) S1PR3GLP1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350015-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2011-08-03 EP disclosed