SCHEMBL3345533

SCHEMBL3345533

Cc1c(C(=O)N[C@H](c2ccc(F)c(F)c2)C2CCC2)c2c([C@@H](c3cc(F)cc(F)c3C(N)=O)C3CCC3)ccc(F)c2c(=O)n1Cc1ncco1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 6/20 0.36
WDR5 P61964 12/20 0.33
PDE2A O00408 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2306426 0.88 CYP2C9 (0.35) S1PR3WDR5
SCHEMBL2306989 0.88 S1PR3 (0.35) S1PR3
SCHEMBL1364240 0.82 S1PR3 (0.42) S1PR3WDR5PDE2A
SCHEMBL2313391 0.79 S1PR3 (0.34) S1PR3
SCHEMBL1364329 0.77 S1PR3 (0.38) S1PR3WDR5
SCHEMBL1366190 0.76 CYP2C9 (0.43) S1PR3WDR5
SCHEMBL2308354 0.76 S1PR3 (0.33) S1PR3
SCHEMBL1364113 0.76 S1PR3 (0.37) S1PR3WDR5
SCHEMBL3380867 0.74 CYP2C9 (0.36) WDR5
SCHEMBL2310390 0.74 CYP2C9 (0.39) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045948-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-04-29 WO disclosed